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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TQ0267 | Endomorphin 1 | Endomorphin-1 | Opioid Receptor |
Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM). | |||
TP1251L | N-terminally acetylated Endomorphin-1 acetate | Ac-L-Tyr-L-Pro-L-Trp-L-Phe-CONH2 | Others |
N-terminally acetylated Endomorphin-1 acetate (Ac-L-Tyr-L-Pro-L-Trp-L-Phe-CONH2) is a modified Endomorphin-1. | |||
TP1251 | N-terminally acetylated Endomorphin-1 | Ac-L-Tyr-L-Pro-L-Trp-L-Phe-CONH2 | |
N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1. | |||
T8991 | BMS986187 | Opioid Receptor | |
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor. | |||
T72423 | Endomorphin 1 acetate | ||
Endomorphin-1 acetate is a highly selective and high-affinity μ-opioid receptor agonist (K i: 1.11 nM) that also demonstrates moderate affinity for kappa 3 binding sites (K i: 20-30 nM). This compound exhibits antinocice... | |||
T26869 | BMS-986122 | BMS 986122 | Opioid Receptor |
BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC5... | |||
T70267 | ADL 08-0011 HCl | ||
ADL 08-0011 is an active metabolite of the μ-opioid receptor antagonist alvimopan. It is produced from alvimopan via amide hydrolysis by gut microbiota. ADL 08-0011 is a μ-opioid receptor antagonist (Ki = 0.25 nM). It is... |